Assay ID | Title | Year | Journal | Article |
AID1745845 | Primary qHTS for Inhibitors of ATXN expression | | | |
AID504810 | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID504812 | Inverse Agonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID651635 | Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression | | | |
AID370883 | Inhibition of human recombinant MMP14 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370869 | Inhibition recombinant MMP1 at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370882 | Inhibition of human recombinant MMP11 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370868 | Activity of human recombinant MMP13 | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370884 | Inhibition of human recombinant MMP15 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370876 | Inhibition of human recombinant MMP3 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370887 | Inhibition of human recombinant ADAMTS5 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370867 | Inhibition recombinant MMP12 at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370877 | Inhibition of human recombinant MMP8 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370631 | Inhibition recombinant MMP3 at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370875 | Inhibition of human recombinant MMP2 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370889 | Inhibition of human recombinant MMP9 by fluorogenic substrate assay | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370879 | Inhibition of human recombinant MMP12 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370878 | Inhibition of human recombinant MMP10 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370874 | Inhibition of human recombinant MMP13 by HxBPyne probe-based competitive activity based protein profiling assay | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370888 | Inhibition of human recombinant MMP8 by fluorogenic substrate assay | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370886 | Inhibition of human recombinant MMP24 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370866 | Inhibition recombinant MMP9 at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370630 | Inhibition recombinant MMP2 at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370873 | Inhibition of human recombinant MMP13 by fluorogenic substrate assay | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
AID370629 | Inhibition of human recombinant MMP13 expressed in Escherichia coli | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370632 | Inhibition recombinant MMP8 expressed in CHO-K1 cells at 100 uM | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate. |
AID370885 | Inhibition of human recombinant MMP16 at 200 uM by HxBPyne probe-based competitive activity based protein profiling assay in presence of 5 uM HxBpane competitor | 2009 | Bioorganic & medicinal chemistry, Feb-01, Volume: 17, Issue:3
| Ranking the selectivity of PubChem screening hits by activity-based protein profiling: MMP13 as a case study. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |